DOLOCAINE

Anesthetics

Description
Shipping Options
Customer Reviews

1. Introduction

DOLOCAINE is a local anesthetic preparation containing Lidocaine Hydrochloride, available in multiple formulations for versatile medical use. It provides rapid, effective local anesthesia for various clinical procedures.

2. Description

Generic Name: Lidocaine HCl
Available Formulations:
- Injection (1%, 2%)
- Topical jelly (2%)
- Cream (5%)
- Spray (10%)
Drug Class: Amide-type local anesthetic

3. Uses

✔ Local anesthesia for minor surgical procedures ✔ Dental anesthesia (infiltration/nerve block) ✔ Cardiac arrhythmias (IV form) ✔ Topical anesthesia for mucous membranes ✔ Post-herpetic neuralgia (patch formulation)

4. Mechanism of Action

Blocks voltage-gated sodium channels
Inhibits depolarization of nerve fibers
Onset: 2-5 minutes (injection), 3-5 minutes (topical)
Duration: 30-120 minutes (varies by formulation)

5. Side Effects

Common:

Injection site reactions (pain, swelling)
Temporary numbness beyond target area
Mild dizziness (systemic absorption)

Serious (Require Immediate Attention):

CNS toxicity (tinnitus, seizures)
Cardiovascular depression
Allergic reactions (rare with amides)

6. Storage

Injection: Room temperature (15-30°C)
Topicals: Below 25°C
Protect from light
Do not freeze

7. Precautions & Warnings

⚠ Contraindications:

Hypersensitivity to amide anesthetics
Severe heart block (for IV use)
Porphyria

⚠ Special Populations:

Elderly: Reduced dose needed
Hepatic impairment: Caution with repeated doses
Pregnancy: Category B (use if benefits outweigh risks)

⚠ Maximum Recommended Doses:

Plain: 4.5 mg/kg (max 300 mg)
With epinephrine: 7 mg/kg (max 500 mg)

8. Comparison of Formulations

Formulation	Concentration	Onset	Duration	Max Dose
Injection	1-2%	2-5 min	30-90 min	4.5 mg/kg
Jelly	2%	3-5 min	15-30 min	3 mg/kg
Spray	10%	1-2 min	10-15 min	3 sprays

9. Clinical Pearls

• Test dose recommended for nerve blocks • Aspirate before injection to avoid IV administration • Add epinephrine (1:200,000) to prolong duration when appropriate • Monitor for CNS symptoms during large dose administration

10. Conclusion

DOLOCAINE remains the gold standard local anesthetic due to its:

Rapid onset
Predictable duration
Excellent safety profile
Multiple formulation options

1. Introduction

2. Description

Generic Name: Lidocaine HCl
Available Formulations:
- Injection (1%, 2%)
- Topical jelly (2%)
- Cream (5%)
- Spray (10%)
Drug Class: Amide-type local anesthetic

3. Uses

✔ Local anesthesia for minor surgical procedures
✔ Dental anesthesia (infiltration/nerve block)
✔ Cardiac arrhythmias (IV form)
✔ Topical anesthesia for mucous membranes
✔ Post-herpetic neuralgia (patch formulation)

4. Mechanism of Action

Blocks voltage-gated sodium channels
Inhibits depolarization of nerve fibers
Onset: 2-5 minutes (injection), 3-5 minutes (topical)
Duration: 30-120 minutes (varies by formulation)

5. Side Effects

Common:

Injection site reactions (pain, swelling)
Temporary numbness beyond target area
Mild dizziness (systemic absorption)

Serious (Require Immediate Attention):

CNS toxicity (tinnitus, seizures)
Cardiovascular depression
Allergic reactions (rare with amides)

6. Storage

Injection: Room temperature (15-30°C)
Topicals: Below 25°C
Protect from light
Do not freeze

7. Precautions & Warnings

⚠ Contraindications:

Hypersensitivity to amide anesthetics
Severe heart block (for IV use)
Porphyria

⚠ Special Populations:

Elderly: Reduced dose needed
Hepatic impairment: Caution with repeated doses
Pregnancy: Category B (use if benefits outweigh risks)

⚠ Maximum Recommended Doses:

Plain: 4.5 mg/kg (max 300 mg)
With epinephrine: 7 mg/kg (max 500 mg)

8. Comparison of Formulations

Formulation	Concentration	Onset	Duration	Max Dose
Injection	1-2%	2-5 min	30-90 min	4.5 mg/kg
Jelly	2%	3-5 min	15-30 min	3 mg/kg
Spray	10%	1-2 min	10-15 min	3 sprays

9. Clinical Pearls

• Test dose recommended for nerve blocks
• Aspirate before injection to avoid IV administration
• Add epinephrine (1:200,000) to prolong duration when appropriate
• Monitor for CNS symptoms during large dose administration

10. Conclusion

DOLOCAINE remains the gold standard local anesthetic due to its:

Rapid onset
Predictable duration
Excellent safety profile
Multiple formulation options

Shipping Options –

We offer a variety of shipping options, including Express Mail Service (EMS), USPS, DHL, FedEx, TNT, UPS, Aramex, Air Cargo, and sea freight.

Terms and Conditions –

Bulk Orders: You are responsible for any local import duties and taxes in your country.

For Patients: When ordering prescription medicines for personal use, or for a friend or relative, a valid medical practitioner’s script or prescription is required.

Return and Refund Policy: Due to the nature of our products, we cannot accept returns or exchanges once a purchase is made. However, in the event of non-delivery, you are eligible for either a 100% refund or a reshipment of your order.

Description
Reviews (0)

1. Introduction

2. Description

Generic Name: Lidocaine HCl
Available Formulations:
- Injection (1%, 2%)
- Topical jelly (2%)
- Cream (5%)
- Spray (10%)
Drug Class: Amide-type local anesthetic

3. Uses

✔ Local anesthesia for minor surgical procedures
✔ Dental anesthesia (infiltration/nerve block)
✔ Cardiac arrhythmias (IV form)
✔ Topical anesthesia for mucous membranes
✔ Post-herpetic neuralgia (patch formulation)

4. Mechanism of Action

Blocks voltage-gated sodium channels
Inhibits depolarization of nerve fibers
Onset: 2-5 minutes (injection), 3-5 minutes (topical)
Duration: 30-120 minutes (varies by formulation)

5. Side Effects

Common:

Injection site reactions (pain, swelling)
Temporary numbness beyond target area
Mild dizziness (systemic absorption)

Serious (Require Immediate Attention):

CNS toxicity (tinnitus, seizures)
Cardiovascular depression
Allergic reactions (rare with amides)

6. Storage

Injection: Room temperature (15-30°C)
Topicals: Below 25°C
Protect from light
Do not freeze

7. Precautions & Warnings

⚠ Contraindications:

Hypersensitivity to amide anesthetics
Severe heart block (for IV use)
Porphyria

⚠ Special Populations:

Elderly: Reduced dose needed
Hepatic impairment: Caution with repeated doses
Pregnancy: Category B (use if benefits outweigh risks)

⚠ Maximum Recommended Doses:

Plain: 4.5 mg/kg (max 300 mg)
With epinephrine: 7 mg/kg (max 500 mg)

8. Comparison of Formulations

Formulation	Concentration	Onset	Duration	Max Dose
Injection	1-2%	2-5 min	30-90 min	4.5 mg/kg
Jelly	2%	3-5 min	15-30 min	3 mg/kg
Spray	10%	1-2 min	10-15 min	3 sprays

9. Clinical Pearls

• Test dose recommended for nerve blocks
• Aspirate before injection to avoid IV administration
• Add epinephrine (1:200,000) to prolong duration when appropriate
• Monitor for CNS symptoms during large dose administration

10. Conclusion

DOLOCAINE remains the gold standard local anesthetic due to its:

Rapid onset
Predictable duration
Excellent safety profile
Multiple formulation options

Reviews

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Description
Reviews (0)

1. Introduction

2. Description

Generic Name: Lidocaine HCl
Available Formulations:
- Injection (1%, 2%)
- Topical jelly (2%)
- Cream (5%)
- Spray (10%)
Drug Class: Amide-type local anesthetic

3. Uses

✔ Local anesthesia for minor surgical procedures
✔ Dental anesthesia (infiltration/nerve block)
✔ Cardiac arrhythmias (IV form)
✔ Topical anesthesia for mucous membranes
✔ Post-herpetic neuralgia (patch formulation)

4. Mechanism of Action

Blocks voltage-gated sodium channels
Inhibits depolarization of nerve fibers
Onset: 2-5 minutes (injection), 3-5 minutes (topical)
Duration: 30-120 minutes (varies by formulation)

5. Side Effects

Common:

Injection site reactions (pain, swelling)
Temporary numbness beyond target area
Mild dizziness (systemic absorption)

Serious (Require Immediate Attention):

CNS toxicity (tinnitus, seizures)
Cardiovascular depression
Allergic reactions (rare with amides)

6. Storage

Injection: Room temperature (15-30°C)
Topicals: Below 25°C
Protect from light
Do not freeze

7. Precautions & Warnings

⚠ Contraindications:

Hypersensitivity to amide anesthetics
Severe heart block (for IV use)
Porphyria

⚠ Special Populations:

Elderly: Reduced dose needed
Hepatic impairment: Caution with repeated doses
Pregnancy: Category B (use if benefits outweigh risks)

⚠ Maximum Recommended Doses:

Plain: 4.5 mg/kg (max 300 mg)
With epinephrine: 7 mg/kg (max 500 mg)

8. Comparison of Formulations

Formulation	Concentration	Onset	Duration	Max Dose
Injection	1-2%	2-5 min	30-90 min	4.5 mg/kg
Jelly	2%	3-5 min	15-30 min	3 mg/kg
Spray	10%	1-2 min	10-15 min	3 sprays

9. Clinical Pearls

• Test dose recommended for nerve blocks
• Aspirate before injection to avoid IV administration
• Add epinephrine (1:200,000) to prolong duration when appropriate
• Monitor for CNS symptoms during large dose administration

10. Conclusion

DOLOCAINE remains the gold standard local anesthetic due to its:

Rapid onset
Predictable duration
Excellent safety profile
Multiple formulation options

Reviews

There are no reviews yet.

Be the first to review “DOLOCAINE”

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